Microwave-assis synthesis of pyrazolo[1,5c] quinazolines and their derivatives

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Date

2014

Journal Title

Journal ISSN

Volume Title

Publisher

Elsevier

Abstract

Microwave accelerated and expedited cyclocondensation reactions of 2-(3-aryl-1H-pyrazol-5-yl)anilines (4) with diverse aryl aldehydes/triethyl orthoformate in water/MeCN (route D) and internal cyclocondensation and aromatization of 5-(2-aminophenyl)-4,5-dihydro-3-arylpyrazole-1-carbaldehyde (7) under MeOH (route E) for the synthesis of a series of pyrazolo[1,5-c]quinazolines and their derivatives (1a–1q) are reported.

Description

Keywords

Microwave heating, Pyrazolo[1,5-c]quinazolines and their derivatives, Cyclocondensation, SynthesisAryl aldehydes

Citation

Kumar, Deependra and Kumar, Raj (2014) Microwave-assis synthesis of pyrazolo[1,5c] quinazolines and their derivatives. Tetrahedron Letters. Vol. 55(16), PP. 2679-2683